31.12.2010   

EN

Official Journal of the European Union

L 348/36


REGULATION (EU) No 1238/2010 OF THE EUROPEAN PARLIAMENT AND OF THE COUNCIL

of 15 December 2010

amending Annex I to Council Regulation (EEC) No 2658/87 as regards the provision of duty-free treatment for specified pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organization and specified products used for the manufacture of finished pharmaceuticals

THE EUROPEAN PARLIAMENT AND THE COUNCIL OF THE EUROPEAN UNION,

Having regard to the Treaty on the Functioning of the European Union, and in particular Article 207 thereof,

Having regard to the proposal from the European Commission,

After transmission of the draft legislative act to the national parliaments,

Acting in accordance with the ordinary legislative procedure (1),

Whereas:

(1)

In the course of the Uruguay Round negotiations, the Community and a number of countries agreed that duty-free treatment should be granted to pharmaceutical products falling within the Harmonised System (HS) Chapter 30 and HS headings 2936, 2937, 2939 and 2941 as well as to designated pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organization, specified salts, esters and hydrates of such INNs, and designated pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals.

(2)

The results of the discussions, as set out in the Record of Discussions, were incorporated into the tariff schedules of the participants annexed to the Marrakesh Protocol to the General Agreement on Tariffs and Trade (GATT) 1994.

(3)

Participants concluded that representatives of World Trade Organization (WTO) members, party to the Record of Discussions, would meet under the auspices of the Council for Trade in Goods of the WTO, normally at least once every three years, to review the product coverage with a view to including, by consensus, additional pharmaceutical products for tariff elimination.

(4)

Three such reviews have taken place with the result that a certain number of additional INNs and pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals have been granted duty-free treatment, that some of those intermediates have been transferred to the list of INNs, and that the list of specified prefixes and suffixes for salts, esters or hydrates of INNs has been expanded.

(5)

A fourth review was deemed appropriate and was launched in 2009. It concluded that a certain number of additional INNs and pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals should be granted duty-free treatment, that some of those intermediates already included in the pharmaceutical sectoral arrangement and its revisions should be transferred to the list of INNs, and that the list of specified prefixes and suffixes for salts, esters or hydrates of INNs should be expanded.

(6)

Council Regulation (EEC) No 2658/87 of 23 July 1987 on the tariff and statistical nomenclature and on the Common Customs Tariff (2) established the Combined Nomenclature (CN) and set out the conventional duty rates of the Common Customs Tariff.

(7)

Regulation (EEC) No 2658/87 should therefore be amended accordingly.

(8)

In order to ensure that the measures provided for in this Regulation apply from 1 January 2011, it should enter into force on the day following that of its publication,

HAVE ADOPTED THIS REGULATION:

Article 1

Annexes 3, 4 and 6 of Section II of Part Three of Annex I to Regulation (EEC) No 2658/87 (Lists of pharmaceutical substances which qualify for duty-free treatment) are hereby amended as follows:

1.

As from 1 January 2011 the Union shall extend duty-free treatment to the INNs listed in Annex I.

2.

As from 1 January 2011 the list of prefixes and suffixes which, in combination with the INNs included in the pharmaceutical sectoral arrangement and its revisions, describe the salts, esters or hydrates of INNs which are also eligible for duty-free treatment, on condition that they are classifiable in the same six-digit HS subheading as the corresponding INN, shall be amended as set out in Annex II.

3.

As from 1 January 2011 the Union shall extend duty-free treatment to the pharmaceutical intermediates used in the production and manufacture of finished pharmaceuticals, listed in Annex III.

4.

As from 1 January 2011 the pharmaceutical intermediates listed in Annex IV shall be withdrawn from the list of such compounds receiving duty-free treatment.

Article 2

This Regulation shall enter into force on the day following that of its publication in the Official Journal of the European Union.

It shall apply from 1 January 2011.

This Regulation shall be binding in its entirety and directly applicable in all Member States.

Done at Strasbourg, 15 December 2010.

For the European Parliament

The President

J. BUZEK

For the Council

The President

O. CHASTEL


(1)  Position of the European Parliament of 23 November 2010 (not yet published in the Official Journal) and decision of the Council of 10 December 2010.

(2)   OJ L 256, 7.9.1987, p. 1.


ANNEX I

List of international non-proprietary names (INNs) to be added to the list of products receiving duty-free treatment included in Annex 3 to Annex I to Regulation (EEC) No 2658/87

CN code

CAS RN

Name

2842 90 80

119175-48-3

fermagate

2843 90 90

759457-82-4

padeliporfin

2844 40 30

123748-56-1

iodofiltic acid (

Formula

)

2904 10 00

21668-77-9

eprodisate

2906 19 00

199798-84-0

elocalcitol

2909 30 90

24150-24-1

terameprocol

2916 19 95

81485-25-8

peretinoin

2916 39 00

51543-40-9

tarenflurbil

2918 19 98

174022-42-5

bevirimat

2919 90 00

258516-89-1

fospropofol

2920 90 85

163133-43-5

naproxcinod

2921 19 99

3687-18-1

tramiprosate

2922 19 85

68392-35-8

afimoxifene

2922 19 85

753449-67-1

ronacaleret

2922 29 00

433265-65-7

faxeladol

2922 50 00

121524-08-1

amibegron

2922 50 00

329773-35-5

cinaciguat

2922 50 00

643094-49-9

fasobegron

2923 10 00

856676-23-8

choline fenofibrate

2924 29 98

847353-30-4

arbaclofen placarbil

2924 29 98

194785-19-8

bedoradrine

2924 29 98

194085-75-1

carisbamate

2924 29 98

254750-02-2

emricasan

2924 29 98

355129-15-6

eprotirome

2924 29 98

402567-16-2

firategrast

2924 29 98

478296-72-9

gabapentin enacarbil

2924 29 98

15866-90-7

incyclinide

2924 29 98

202844-10-8

indantadol

2924 29 98

96847-55-1

levomilnacipran

2924 29 98

608137-32-2

lisdexamfetamine

2924 29 98

652990-07-3

milveterol

2924 29 98

181816-48-8

ombrabulin

2924 29 98

289656-45-7

senicapoc

2925 19 95

19171-19-8

pomalidomide

2928 00 90

22033-87-0

olesoxime

2928 00 90

2675-35-6

sivifene

2928 00 90

816458-31-8

tecovirimat

2928 00 90

238750-77-1

tosedostat

2928 00 90

149647-78-9

vorinostat

2929 90 00

31645-39-3

palifosfamide

2930 90 99

608141-41-9

apremilast

2930 90 99

216167-92-9

camobucol

2930 90 99

211513-37-0

dalcetrapib

2930 90 99

69819-86-9

darinaparsin

2930 90 99

488832-69-5

elesclomol

2930 90 99

216167-95-2

elsibucol

2930 90 99

168682-53-9

ezatiostat

2930 90 99

58569-55-4

metenkefalin

2930 90 99

887148-69-8

monepantel

2930 90 99

603139-19-1

odanacatib

2930 90 99

162520-00-5

salirasib

2930 90 99

216167-82-7

succinobucol

2930 90 99

125961-82-2

tipelukast

2931 00 99

125973-56-0

amsilarotene

2932 19 00

253128-41-5

eribulin

2932 19 00

186953-56-0

pafuramidine

2932 29 85

195883-06-8

omtriptolide

2932 99 00

664338-39-0

arterolane

2932 99 00

183133-96-2

cabazitaxel

2932 99 00

401925-43-7

celivarone

2932 99 00

461432-26-8

dapagliflozin

2932 99 00

118457-15-1

dexnebivolol

2932 99 00

156294-36-9

larotaxel

2932 99 00

118457-16-2

levonebivolol

2932 99 00

83461-56-7

mifamurtide

2932 99 00

117570-53-3

vadimezan

2933 19 90

496775-61-2

eltrombopag

2933 19 90

206884-98-2

niraxostat

2933 19 90

410528-02-8

palovarotene

2933 19 90

376592-42-6

totrombopag

2933 29 90

183659-72-5

catramilast

2933 29 90

944263-65-4

demiditraz

2933 29 90

867153-61-5

dulanermin

2933 29 90

320367-13-3

lixisenatide

2933 29 90

698389-00-3

rolipoltide

2933 29 90

697766-75-9

velafermin

2933 39 99

147084-10-4

alcaftadine

2933 39 99

54-96-6

amifampridine

2933 39 99

249921-19-5

anamorelin

2933 39 99

319460-85-0

axitinib

2933 39 99

208110-64-9

befiradol

2933 39 99

330942-05-7

betrixaban

2933 39 99

201034-75-5

daporinad

2933 39 99

209783-80-2

entinostat

2933 39 99

412950-27-7

goxalapladib

2933 39 99

218791-21-0

imisopasem manganese

2933 39 99

103129-82-4

levamlodipine

2933 39 99

154357-42-3

levonadifloxacin

2933 39 99

108147-54-2

migalastat

2933 39 99

453562-69-1

motesanib

2933 39 99

139145-27-0

parogrelil

2933 39 99

459856-18-9

pexacerfont

2933 39 99

706779-91-1

pimavanserin

2933 39 99

362665-56-3

pitolisant

2933 39 99

861151-12-4

rosonabant

2933 39 99

701977-09-5

taranabant

2933 39 99

189950-11-6

tropantiol

2933 39 99

793655-64-8

vapitadine

2933 39 99

139290-65-6

volinaserin

2933 49 90

141388-76-3

besifloxacin

2933 49 90

697761-98-1

elvitegravir

2933 49 90

185055-67-8

ferroquine

2933 49 90

445041-75-8

intiquinatine

2933 49 90

378746-64-6

nemonoxacin

2933 49 90

245765-41-7

ozenoxacin

2933 49 90

412950-08-4

rilapladib

2933 49 90

871224-64-5

almorexant

2933 49 90

863029-99-6

balamapimod

2933 49 90

698387-09-6

neratinib

2933 49 90

154652-83-2

tezampanel

2933 49 90

128253-31-6

veliflapon

2933 59 95

791828-58-5

aderbasib

2933 59 95

840486-93-3

adipiplon

2933 59 95

850649-61-5

alogliptin

2933 59 95

859212-16-1

bafetinib

2933 59 95

380843-75-4

bosutinib

2933 59 95

839712-12-8

cariprazine

2933 59 95

414910-27-3

casopitant

2933 59 95

288383-20-0

cediranib

2933 59 95

849550-05-6

cevipabulin

2933 59 95

827318-97-8

danusertib

2933 59 95

356057-34-6

darapladib

2933 59 95

501000-36-8

dutacatib

2933 59 95

247257-48-3

fimasartan

2933 59 95

3432-99-3

folitixorin

2933 59 95

668270-12-0

linagliptin

2933 59 95

441798-33-0

macitentan

2933 59 95

641571-10-0

nilotinib

2933 59 95

763113-22-0

olaparib

2933 59 95

686344-29-6

otenabant

2933 59 95

625115-55-1

riociguat

2933 59 95

486460-32-6

sitagliptin

2933 59 95

425637-18-9

sotrastaurin

2933 59 95

309913-83-5

talmapimod

2933 59 95

113857-87-7

talotrexin

2933 59 95

274693-27-5

ticagrelor

2933 59 95

306296-47-9

vicriviroc

2933 69 80

775351-65-0

imeglimin

2933 79 00

461443-59-4

aplaviroc

2933 79 00

189691-06-3

bremelanotide

2933 79 00

813452-18-5

carmegliptin

2933 79 00

405169-16-6

dovitinib

2933 79 00

536748-46-6

eribaxaban

2933 79 00

473289-62-2

ilepatril

2933 79 00

180694-97-7

mimopezil

2933 79 00

579475-18-6

orvepitant

2933 79 00

449811-01-2

pamapimod

2933 79 00

248282-01-1

paquinimod

2933 79 00

380917-97-5

perampanel

2933 79 00

552292-08-7

rolapitant

2933 79 00

425386-60-3

semagacestat

2933 79 00

515814-01-4

voclosporin

2933 99 80

481629-87-2

aleplasinin

2933 99 80

394730-60-0

boceprevir

2933 99 80

649735-63-7

brivanib alaninate

2933 99 80

483369-58-0

denagliptin

2933 99 80

284019-34-7

denibulin

2933 99 80

481631-45-2

diaplasinin

2933 99 80

272105-42-7

disitertide

2933 99 80

227318-71-0

epetirimod

2933 99 80

259793-96-9

favipiravir

2933 99 80

871576-03-3

flovagatran

2933 99 80

229305-39-9

golotimod

2933 99 80

258818-34-7

larazotide

2933 99 80

571170-77-9

laropiprant

2933 99 80

616202-92-7

lorcaserin

2933 99 80

868771-57-7

melogliptin

2933 99 80

803712-67-6

obatoclax

2933 99 80

404950-80-7

panobinostat

2933 99 80

625114-41-2

piragliatin

2933 99 80

74847-35-1

pyronaridine

2933 99 80

872178-65-9

rabeximod

2933 99 80

355151-12-1

rotigaptide

2933 99 80

497221-38-2

rusalatide

2933 99 80

187602-11-5

sofigatran

2933 99 80

227318-75-4

sotirimod

2933 99 80

402957-28-2

telaprevir

2933 99 80

848084-83-3

tigapotide

2933 99 80

393105-53-8

tiplasinin

2933 99 80

620948-93-8

vabicaserin

2933 99 80

794466-70-9

vernakalant

2934 10 00

544417-40-5

capadenoson

2934 10 00

302962-49-8

dasatinib

2934 10 00

223132-37-4

inolitazone

2934 10 00

241479-67-4

isavuconazole

2934 10 00

338990-84-4

isavuconazonium chloride

2934 10 00

607723-33-1

lobeglitazone

2934 10 00

280782-97-0

managlinat dialanetil

2934 10 00

790299-79-5

masitinib

2934 10 00

223673-61-8

mirabegron

2934 10 00

501948-05-6

rosabulin

2934 10 00

447406-78-2

sodelglitazar

2934 10 00

760937-92-6

teneligliptin

2934 20 80

848344-36-5

bentamapimod

2934 20 80

870093-23-5

talarozole

2934 99 90

320345-99-1

aclidinium bromide

2934 99 90

222551-17-9

adoprazine

2934 99 90

207623-20-9

agatolimod

2934 99 90

475479-34-6

aleglitazar

2934 99 90

870524-46-2

amolimogene bepiplasmid

2934 99 90

875446-37-0

anacetrapib

2934 99 90

250386-15-3

apadenoson

2934 99 90

541550-19-0

apilimod

2934 99 90

160707-69-7

apricitabine

2934 99 90

147403-03-0

azilsartan

2934 99 90

863031-21-4

azilsartan medoxomil

2934 99 90

757942-43-1

bederocin

2934 99 90

627861-07-8

beperminogene perplasmid

2934 99 90

959961-96-7

bevasiranib

2934 99 90

769901-96-4

capeserod

2934 99 90

868540-17-4

carfilzomib

2934 99 90

872847-66-0

cenersen

2934 99 90

80295-38-1

conestat alfa

2934 99 90

903916-27-8

custirsen

2934 99 90

187865-22-1

derquantel

2934 99 90

134379-77-4

dexelvucitabine

2934 99 90

247046-52-2

dilopetine

2934 99 90

480449-70-5

edoxaban

2934 99 90

188181-42-2

elacytarabine

2934 99 90

98819-76-2

esreboxetine

2934 99 90

763903-67-9

fosalvudine tidoxil

2934 99 90

172673-20-0

fosaprepitant

2934 99 90

522664-63-7

ibodutant

2934 99 90

405159-59-3

idrabiotaparinux sodium

2934 99 90

188116-07-6

imepitoin

2934 99 90

335619-18-6

inakalant

2934 99 90

1391-36-2

lancovutide

2934 99 90

189059-71-0

lapaquistat

2934 99 90

327026-93-7

lensiprazine

2934 99 90

170632-47-0

lificiguat

2934 99 90

852313-25-8

litenimod

2934 99 90

1000120-98-8

mipomersen

2934 99 90

62253-63-8

nepidermin

2934 99 90

26833-87-4

omacetaxine mepesuccinate

2934 99 90

269718-84-5

pardoprunox

2934 99 90

219923-85-0

pramiconazole

2934 99 90

377727-87-2

preladenant

2934 99 90

524684-52-4

prinaberel

2934 99 90

865311-47-3

quarfloxin

2934 99 90

869884-78-6

radezolid

2934 99 90

496054-87-6

radiprodil

2934 99 90

518048-05-0

raltegravir

2934 99 90

787548-03-2

regrelor

2934 99 90

820957-38-8

retosiban

2934 99 90

572924-54-0

ridaforolimus

2934 99 90

128517-07-7

romidepsin

2934 99 90

93265-81-7

ropidoxuridine

2934 99 90

151823-14-2

sapacitabine

2934 99 90

379231-04-6

saracatinib

2934 99 90

791635-59-1

simotaxel

2934 99 90

119567-79-2

taribavirin

2934 99 90

332012-40-5

telatinib

2934 99 90

925681-61-4

trabedersen

2934 99 90

189003-92-7

trelanserin

2934 99 90

296251-72-4

velimogene aliplasmid

2934 99 90

904302-98-3

viquidacin

2934 99 90

872525-61-6

votucalis

2934 99 90

221877-54-9

zotarolimus

2935 00 90

197904-84-0

apricoxib

2935 00 90

769169-27-9

begacestat

2935 00 90

414864-00-9

belinostat

2935 00 90

313682-08-5

brecanavir

2935 00 90

839673-52-8

cevoglitazar

2935 00 90

358970-97-5

drinabant

2935 00 90

865200-20-0

giripladib

2935 00 90

464213-10-3

ibipinabant

2935 00 90

173424-77-6

laromustine

2935 00 90

398507-55-6

lodenafil carbonate

2935 00 90

136564-68-6

masilukast

2935 00 90

170569-88-7

mavacoxib

2935 00 90

862189-95-5

mirodenafil

2935 00 90

439687-69-1

nelivaptan

2935 00 90

691852-58-1

nesbuvir

2935 00 90

778576-62-8

oglemilast

2935 00 90

444731-52-6

pazopanib

2935 00 90

362505-84-8

relacatib

2935 00 90

243984-11-4

resatorvid

2935 00 90

519055-62-0

tasisulam

2935 00 90

186497-07-4

zibotentan

2936 29 00

104121-92-8

eldecalcitol

2936 29 00

31690-09-2

levomefolic acid

2937 19 00

782500-75-8

albiglutide

2937 19 00

348119-84-6

obinepitide

2937 19 00

295350-45-7

ozarelix

2937 19 00

275371-94-3

taspoglutide

2937 19 00

218949-48-5

tesamorelin

2937 19 00

22006-64-0

tridecactide

2937 22 00

132245-57-9

dexamethasone cipecilate

2937 22 00

397864-44-7

fluticasone furoate

2937 29 00

211254-73-8

lonaprisan

2937 50 00

333963-42-1

cobiprostone

2937 50 00

172740-14-6

posaraprost

2937 90 00

834153-87-6

elagolix

2937 90 00

609799-22-6

tasimelteon

2937 90 00

342577-38-2

velneperit

2939 19 00

73232-52-7

methylnaltrexone bromide

2939 59 00

136199-02-5

rolofylline

2939 99 00

850607-58-8

darotropium bromide

2939 99 00

187852-63-7

delimotecan

2940 00 00

9007-72-1

ferric carboxymaltose

2940 00 00

442201-24-3

remogliflozin etabonate

2940 00 00

408504-26-7

sergliflozin etabonate

2941 90 00

467214-20-6

alvespimycin

2941 90 00

677017-23-1

berubicin

2941 90 00

229016-73-3

ceftaroline fosamil

2941 90 00

318498-76-9

flopristin

2941 90 00

145435-72-9

gamithromycin

2941 90 00

325965-23-9

linopristin

2941 90 00

857402-23-4

retaspimycin

2941 90 00

305841-29-6

sagopilone

2941 90 00

75747-14-7

tanespimycin

2941 90 00

328898-40-4

tildipirosin

2941 90 00

222400-20-6

tomopenem

2941 90 00

63409-12-1

tylvalosin

3001 90 91

9041-08-1

semuloparin sodium

3002 10 91

792921-10-9

abagovomab

3002 10 91

910649-32-0

anrukinzumab

3002 10 91

648904-28-3

bavituximab

3002 10 91

402710-27-4

(light chain)

402710-25-2

(heavy chain)

canakinumab

3002 10 99

945228-49-9

citatuzumab bogatox

3002 10 91

880486-59-9

dacetuzumab

3002 10 91

615258-40-7

denosumab

3002 10 91

762260-74-2

efungumab

3002 10 91

89957-37-9

gantenerumab

3002 10 91

680188-33-4

ibalizumab

3002 10 91

477202-00-9

ipilimumab

3002 10 91

640735-09-7

iratumumab

3002 10 91

845816-02-6

lexatumumab

3002 10 91

903512-50-5

lucatumumab

3002 10 91

899796-83-9

milatuzumab

3002 10 91

677010-34-3

motavizumab

3002 10 91

676258-98-3

naptumomab estafenatox

3002 10 91

828933-51-3

nimotuzumab

3002 10 91

949142-50-1

obinutuzumab

3002 10 91

637334-45-3

ocrelizumab

3002 10 91

881191-44-2

otelixizumab

3002 10 91

372075-37-1

sontuzumab

3002 10 91

705287-60-1

stamulumab

3002 10 91

339086-80-5

tadocizumab

3002 10 91

592557-43-2

(light chain)

592557-41-0

(heavy chain)

tenatumomab

3002 10 91

876387-05-2

teplizumab

3002 10 91

918127-53-4

tigatuzumab

3002 10 91

745013-59-6

tremelimumab

3002 10 91

339986-90-2

tucotuzumab celmoleukin

3002 10 91

728917-18-8

veltuzumab

3002 10 91

896731-82-1

conatumumab

3002 10 91

892553-42-3

etaracizumab

3002 10 91

944548-38-3

foravirumab

3002 10 91

944548-37-2

rafivirumab

3002 10 91

880266-57-9

tanezumab

3002 10 91

815610-63-0

ustekinumab

3002 10 95

862111-32-8

aflibercept

3002 10 95

845264-92-8

atacicept

3002 10 95

909110-25-4

baminercept

3002 10 95

9001-27-8

beroctocog alfa

3002 10 95

879555-13-2

epoetin kappa

3002 10 95

762263-14-9

epoetin theta

3002 10 95

501081-76-1

rilonacept

3002 10 95

267639-76-9

romiplostim

3002 10 95

869858-13-9

thrombin alfa

3002 10 95

897936-89-9

vatreptacog alfa (activated)

3002 10 95

472960-22-8

albinterferon alfa-2b

3002 10 95

869881-54-9

briobacept

3002 10 95

606138-08-3

catridecacog

3002 10 95

716840-32-3

denenicokin

3002 10 95

931101-84-7

troplasminogen alfa

3002 10 99

934216-54-3

alacizumab pegol

3002 20 00

181477-43-0

disomotide

3002 20 00

181477-91-8

ovemotide

3002 20 00

915019-08-8

tertomotide

3002 20 00

295371-00-5

verpasep caltespen

3002 90 90

473553-86-5

alferminogene tadenovec

3002 90 90

929881-05-0

alipogene tiparvovec

3002 90 90

600735-73-7

contusugene ladenovec

3002 90 90

851199-59-2

linaclotide

3002 90 90

898830-54-1

sitimagene ceradenovec

3002 90 90

721946-42-5

transferrin aldifitox

3507 90 90

9026-00-0

bucelipase alfa

3507 90 90

885051-90-1

pegloticase

3507 90 90

884604-91-5

velaglucerase alfa

3911 90 99

892497-01-7

azoximer bromide


ANNEX II

List of prefixes and suffixes which, in combination with the INNs of Annex 3 to Annex I to Regulation (EEC) No 2658/87, describe the salts, esters or hydrates of INNs; these salts, esters and hydrates are free of duty, on condition that they are classifiable in the same six-digit HS subheading as the corresponding INN

The references to ‘International Nonproprietary Names (INN) for pharmaceutical substances, names for radicals and groups, comprehensive list 2004’ are replaced by ‘International Nonproprietary Names (INN) for pharmaceutical substances, names for radicals, groups and others, comprehensive list 2007’.

The following prefixes or suffixes are added to the list included in Annex 4 to Annex I to Regulation (EEC) No 2658/87:

Preferred prefix or suffix

Synonym

Systematic name when different

alanetil (INNRG)

 

[(S)-1-ethoxy-1-oxo-propan-2-yl]amino (INNCN)

alaninate (INNRG)

 

L-alaninate (INNCN)

alapivoxil (INNRG)

 

L-alanyl, [(2,2-dimethylpropanoyl)oxy]metyl (INNCN)

aldifitox (INNRG)

 

(4-iminobutane-1,4-diyl)sulfanediyl[(3RS)-2,5-dioxopyrrolidine-1,3-diyl]-1,3-phenylenecarbonyl and forming an N-benzoyl derivative of a primary amine group of diphtheria [550-L-phenylalanine]toxin from Corynebacterium diphtheriae-(26-560)-peptide (INNCN)

besudotox (INNRG)

 

L-lysyl-L-alanyl-L-serylglycylglycine (linker) fusion protein with des-(365-380)-[Asn364,Val407,Ser515,Gln590,Gln606,Arg613]exotoxin A (Pseudomonas aeruginosa)-(251-613)-peptide (toxin with region IA and first 16 residues of region IB deleted) (INNCN)

ceribate (INNRG)

 

rac-2,3-dihydroxypropyl carbonate (ester) (INNCN)

cipecilate (INNRG)

 

cyclohexanecarboxylate (ester), cyclopropanecarboxylate (ester) (INNCN)

dalanated (INNRG)

 

des-B30-alanine (INNCN)

enacarbil (INNRG)

 

{rac-1-[(2-methylpropanoyl)oxy]ethoxy}carbonyl (INNCN)

estafenatox (INNRG)

 

glycylglycyl-L-proline (linker) fusion protein with enterotoxin type A (Staphylococcus aureus)-(1-33)-peptidyl-L-seryl[Ser36,Ser37,Glu38,Lys39,Ala41,Thr46,Thr71,Ala72,Ser75,Glu76,Glu78,Ser80,Ser81,Thr214,Ser217,Thr219,Ser220,Ser222,Ser224]enterotoxin type E (Staphylococcus aureus)-(32-230)-peptide (synthetic superantigen SEA/E-120) (INNCN)

etexilate (INNRG)

 

ethyl, (hexyloxy)carbonyl

fosamil (INNRG)

 

phosphono (INNCN)

glucuronide (INNRG)

 

β-D-glucopyranosiduronic acid [oside] (INNCN)

medocaril (INNRG)

 

[(5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy]carbonyl (INNCN)

paptox (INNRG)

 

protein PAP (Phytolacca americana antiviral) (INNCN)

placarbil (INNRG)

 

(R)-2-methyl-1-[(2-methylpropanoyl)oxy]propoxy}carbonyl) (INNCN)

The systematic name of the following prefix or suffix is amended as follows:

Preferred prefix or suffix

Synonym

Systematic name when different

aritox (INNRG)

 

ricin A chain (INNCN)


ANNEX III

List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be added to the list of products receiving duty-free treatment included in Annex 6 to Annex I to Regulation (EEC) No 2658/87

CN code

CAS RN

Name

2843 29 00

22199-08-2

[4-amino-N-(pyrimidin-2(1H)-ylidene-κN1)benzenesulfonamidato-κO]silver

2905 39 95

281214-27-5

(2R,3R)-2,3-dimethylbutane-1,4-diyl bis(4-methylbenzenesulfonate)

2905 59 98

441002-17-1

4-chlorobutyl 2-nitrobenzenesulfonate

2909 30 90

92878-95-0

2-(3-chloropropoxy)-1-methoxy-4-nitrobenzene

2909 30

503070-57-3

2-({2-[(6-bromohexyl)oxy]ethoxy}methyl)-1,3-dichlorobenzene

2909 30

461432-23-5

4-(5-bromo-2-chlorobenzyl)phenyl ethyl ether

2909 49 80

185954-75-0

(3R)-3-methoxydecan-1-ol

2909 49 80

85309-91-7

2-[(2,6-dichlorobenzyl)oxy]ethanol

2909 49 80

160969-03-9

2-[2-(2,2,2-trifluoroethoxy)phenoxy]ethyl methanesulfonate

2909 50 00

167145-13-3

2-[2-(3-methoxyphenyl)ethyl]phenol

2910 20 00

15448-47-2

(2R)-2-methyloxirane

2910 90 00

62600-71-9

(2R)-2-(3-chlorophenyl)oxirane

2910 90 00

702687-42-1

(2R)-2-[(5-bromo-2,3-difluorophenoxy)methyl]oxirane

2910 90 00

683276-64-4

[(2R)-2-methyloxiran-2-yl]methyl 4-nitrobenzenesulfonate

2913 00 00

90035-34-0

4′-(trifluoromethyl)biphenyl-4-carbaldehyde

2914 40 90

17752-16-8

(3β)-3-hydroxycholest-5-en-24-one

2914 50 00

974-23-2

(3β,16α)-3-hydroxy-16,17-epoxypregn-5-en-20-one

2914 70 00

13054-81-4

4-chloro-heptane-3,5-dione

2914 70 00

10226-30-9

6-chlorohexan-2-one

2915 60 90

53064-79-2

iodomethyl pivalate

2915 90 00

22328-90-1

(3R)-3-methylhexanoic acid

2915 90 00

1069-66-5

sodium 2-propylpentanoate

2916 20 00

211515-46-7

1-(2-ethylbutyl)cyclohexanecarbonyl chloride

2916 20 00

381209-09-2

1-(2-ethylbutyl)cyclohexanecarboxylic acid

2916 20 00

7077-05-6

trans-4-(propan-2-yl)cyclohexanecarboxylic acid

2916 39 00

21900-39-0

5-fluoro-2-methylbenzoyl chloride

2916 39 00

17625-03-5

sodium hydrogen 3-sulfonatobenzoate

2917 19 90

76-72-2

diethyl ethyl(pentan-2-yl)propanedioate

2918 29 00

376592-58-4

5′-chloro-2′-hydroxy-3′-nitrobiphenyl-3-carboxylic acid

2918 99 90

709031-28-7

(3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl)(oxo)acetic acid

2918 99 90

35480-52-5

2,5-bis(2,2,2-trifluoroethoxy)benzoic acid

2918 99 90

4651-67-6

(3α,5β)-3-hydroxy-7-oxocholan-24-oic acid

2918 99 90

52179-28-9

ethyl 2-[4-(2,2-dichlorocyclopropyl)phenoxy]-2-methylpropanoate

2918 99 90

530141-60-7

methyl 3-(5-{[4-(cyclopentyloxy)-2-hydroxyphenyl]carbonyl}-2-hydroxyphenyl)propanoate

2920 90 10

91526-18-0

4-(hydroxymethyl)-5-methyl-1,3-dioxol-2-one

2921 49 00

334477-60-0

(1R)-1-[3,5-bis(trifluoromethyl)phenyl]-N-methylethanamine

2921 49 00

376608-71-8

(1R,2S)-2-(3,4-difluorophenyl)cyclopropanaminium (2R)-hydroxy(phenyl)ethanoate

2921 49 00

1034457-07-2

2-(2,3-dihydro-1H-inden-2-yl)propan-2-amine hydrochloride

2921 49 00

945717-05-5

2-(4-chloro-3-ethylphenyl)ethanamine hydrochloride

2921 49 00

89-97-4

2-chlorobenzylamine

2921 49 00

945717-43-1

N-(4-tert-butylbenzyl)-2-(4-chloro-3-ethylphenyl)ethanamine

2921 51 90

150812-21-8

N4-[(4-fluorophenyl)methyl]-2-nitro-1,4-benzenediamine

2922 19 85

1035455-90-3

(2R)-1-(5-bromo-2,3-difluorophenoxy)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}propan-2-ol hydrochloride

2922 19 85

0-00-0

[2-(chloromethyl)-4-(dibenzylamino)phenyl]methanol hydrochloride

2922 19 85

133-51-7

antimonic acid – 1-deoxy-1-(methylamino)-D-glucitol (1:1)

2922 19 85

1035455-87-8

ethyl (2E)-3-(3-{[(2R)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}-2-hydroxypropyl]oxy}-4,5-difluorophenyl)prop-2-enoate hydrochloride

2922 19 85

702686-97-3

ethyl 3-(3-{[(2R)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}-2-hydroxypropyl]oxy}-4,5-difluorophenyl)propanoate hydrochloride

2922 29 00

20059-73-8

2-[4-(aminomethyl)phenoxy]-N,N-dimethylethanamine

2922 49 85

848133-35-7

(2E)-4-(dimethylamino)but-2-enoic acid hydrochloride

2922 49 85

610300-07-7

(3S,5R)-3-amino-5-methyloctanoic acid

2922 49 85

610300-00-0

(3S,5R)-3-amino-5-methyloctanoic acid hydrochloride

2922 49 85

143785-86-8

4-(1-aminocyclopropyl)-2,3,5-trifluorobenzoic acid

2922 49 85

848949-85-9

4-fluoro-L-leucine – ethyl hydrogen sulfate (1:1)

2922 49 85

39068-93-4

methyl 2-(dimethylamino)-2-phenylbutanoate

2922 49 85

168619-25-8

methyl 3′-aminobiphenyl-3-carboxylate

2922 49 85

82834-12-6

N-[(2S)-1-ethoxy-1-oxopentan-2-yl]-L-alanine

2922 49 85

94133-84-3

sodium 2-amino-2-phenylbutanoate

2922 50 00

503070-58-4

triphenylacetic acid – 4-{(1R)-2-[(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl)amino]-1-hydroxyethyl}-2-(hydroxymethyl)phenol (1:1)

2924 19 00

62009-47-6

2-aminomalonamide

2924 19 00

7355-58-0

N-(2-chloroethyl)acetamide

2924 29 98

361442-00-4

{2-[(tert-butoxycarbonyl)amino]-3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl}acetic acid

2924 29 98

266993-72-0

2,3-diaminobenzamide dihydrochloride

2924 29 98

168080-49-7

2-chloro-4-{[(5-fluoro-2-methylphenyl)carbonyl]amino}benzoic acid

2924 29 98

317374-08-6

2-methyl-4-{[(2-methylphenyl)carbonyl]amino}benzoic acid

2924 29 98

143785-84-6

4-(1-carbamoylcyclopropyl)-2,3,5-trifluorobenzoic acid

2924 29 98

143785-87-9

4-[1-(acetylamino)cyclopropyl]-2,3,5-trifluorobenzoic acid

2924 29 98

108166-22-9

4-{[(2-methylphenyl)carbonyl]amino}benzoic acid

2924 29 98

150812-23-0

ethyl {4-[(4-fluorobenzyl)amino]-2-nitrophenyl}carbamate

2924 29 98

22316-45-6

ethyl 3-[(5-chloro-2-nitrophenyl)(phenyl)amino]-3-oxopropanoate

2924 29 98

316173-29-2

methyl (1S,2S,3S,4R)-3-[(1S)-1-amino-2-ethylbutyl]-4-[(tert-butoxycarbonyl)amino]-2-hydroxycyclopentanecarboxylate

2924 29 98

1142-20-7

N-benzyloxycarbonyl-L-alanine

2924 29 98

84996-93-0

N-cyclohexyl-5-hydroxypentanamide

2924 29 98

579494-66-9

propyl {4-[2-(diethylamino)-2-oxoethoxy]-3-ethoxyphenyl}acetate

2925 19 95

265136-65-0

ethyl 3-amino-4-[2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethoxy]but-2-enoate

2926 90 95

855425-38-6

1-(2-ethylbutyl)cyclohexanecarbonitrile

2926 90 95

846023-24-3

2-cyano-N-(2,4-dichloro-5-methoxyphenyl)acetamide

2926 90 95

591769-05-0

3-cyclopentylprop-2-enenitrile

2926 90 95

20099-89-2

4-(bromoacetyl)benzonitrile

2926 90 95

474554-45-5

4,5-diethoxy-3-fluorobenzene-1,2-dicarbonitrile

2926 90 95

79370-78-8

5-hydroxybenzene-1,3-dicarbonitrile

2926 90 95

139481-28-0

methyl 2-{[(2′-cyanobiphenyl-4-yl)methyl]amino}-3-nitrobenzoate

2928 00 90

860035-10-5

1-({[(2,5-dioxopyrrolidin-1-yl)oxy]carbonyl}oxy)ethyl 2-methylpropanoate

2928 00 90

910656-45-0

2-hydroxy-2-(trifluoromethyl)butanehydrazide

2928 00 90

95759-10-7

4-chloro-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoic acid

2928 00 90

473927-63-8

ethyl (2Z)-chloro[2-(4-methoxyphenyl)hydrazinylidene]ethanoate

2928 00 90

158671-29-5

N,2-dihydroxy-4-methylbenzamide

2928 00 90

84080-68-2

tert-butyl (2Z)-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoate

2928 00 90

268544-50-9

tert-butyl-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoate

2930 90 99

13459-62-6

{2-[(4-chlorophenyl)sulfanyl]phenyl}acetic acid

2930 90 99

211513-21-2

1-(2-ethylbutyl)-N-(2-sulfanylphenyl)cyclohexanecarboxamide

2930 90 99

860035-07-0

1-{[(methylsulfanyl)carbonyl]oxy}ethyl 2-methylpropanoate

2930 90 99

893407-18-6

2,2,2-trifluoro-1-[4′-(methylsulfonyl)biphenyl-4-yl]ethanone

2930 90 99

60759-00-4

3,4-diethoxybenzenecarbothioamide

2930 90 99

21048-05-5

N-methylbenzenecarbothiohydrazide

2931 00 99

13682-94-5

(2-bromoethenyl)(trimethyl)silane

2931 00 99

914922-89-7

(2R,4R)-4-[[(1,1-dimethylethyl)dimethylsilyl]oxy]-N-methoxy-N,2-dimethyl-7-oxoheptanamide

2931 00 99

914922-88-6

(2R,4R)-4-{[tert-butyl(dimethyl)silyl]oxy}-N-methoxy-N,2-dimethyloct-7-enamide

2931 00 99

871355-80-5

(4R)-2-bromo-7-{[tert-butyl(diphenyl)silyl]oxy}hept-1-en-4-yl 4-methylbenzenesulfonate

2931 00 99

89694-48-4

(5-chloro-2-methoxyphenyl)boronic acid

2931 00 99

701278-08-2

[(1R,5S)-5-[dimethyl(phenyl)silyl]-2-{[(2-methoxypropan-2-yl)oxy]methyl}cyclopent-2-en-1-yl]methanol

2931 00 99

701278-09-3

{(4S,5R)-5-[(benzyloxy)methyl]-4-[dimethyl(phenyl)silyl]cyclopent-1-en-1-yl}methanol

2931 00 99

796967-18-5

1-(2-fluoro-5-methylphenyl)-3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]urea

2931 00 99

172732-52-4

2-(1,3,2-dioxaborinan-2-yl)benzonitrile

2931 00 99

185411-12-5

methyl 3-(trimethylsilyl)pent-4-enoate

2932 19 00

253128-10-8

(1S)-1,5:7,10-dianhydro-12,13-bis-O-[tert-butyl(dimethyl)silyl]-2,3,4,6,8,11-hexadeoxy-1-{2-[(2S,5S)-5-(3-hydroxypropyl)-3-methylidenetetrahydrofuran-2-yl]ethyl}-3-methyl-9-O-methyl-4-methylidene-8-[(phenylsulfonyl)methyl]-D-arabino-D-altro-tridecitol

2932 19 00

441045-17-6

(1S,3S,6S,9S,12S,14R,16R,18S,20R,21R,22S,26R,29S,31R,32S,33R,35R,36S)-20-[(2S)-3-amino-2-hydroxypropyl]-21-methoxy-14-methyl-8,15-bis(methylene)-2,19,30,34,37,39,40,41-octaoxanonacyclo[24.9.2.13,32.13,33.16,9.112,16.018,22.029,36.031,35]hentetracontan-24-one methanesulfonate

2932 29 85

916069-80-2

(4S)-4-(fluoromethyl)dihydrofuran-2(3H)-one

2932 29 85

63106-93-4

1-phenyl-3-oxabicyclo[3.1.0]hexan-2-one

2932 29 85

7734-80-7

2-oxo-2H-chromene-6-carboxylic acid

2932 29 85

0-00-0

4-(4-fluorophenyl)-7-(isothiocyanatomethyl)-2H-chromen-2-one

2932 29 85

947408-91-5

6-[(2,4-dihydroxyphenyl)carbonyl]-2H-chromen-2-one

2932 29 85

947408-90-4

6-[(2,4-dimethoxyphenyl)carbonyl]-2H-chromen-2-one

2932 99 00

452342-08-4

(1R)-2-(benzylamino)-1-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)ethanol

2932 99 00

99541-23-8

(1R,2S,3R,4R,5R)-4-azido-2-{[(4aR,6S,7R,8S,8aR)-7,8-bis(benzyloxy)-2-phenylhexahydropyrano[3,2-d][1,3]dioxin-6-yl]oxy}-6,8-dioxabicyclo[3.2.1]oct-3-yl acetate

2932 99 00

461432-25-7

(1S)-2,3,4,6-tetra-O-acetyl-1,5-anhydro-1-[4-chloro-3-(4-ethoxybenzyl)phenyl]-D-glucitol

2932 99 00

196597-79-2

(2E)-1,2,6,7-tetrahydro-8H-indeno[5,4-b]furan-8-ylideneethanenitrile

2932 99 00

3308-94-9

2-(3-chloropropyl)-2-(4-fluorophenyl)-1,3-dioxolane

2932 99 00

274693-53-7

[(3aS,4R,6S,6aR)-6-hydroxy-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl]carbamate

2932 99 00

185954-98-7

[6(2Z,3R)]-3-O-decyl-2-deoxy-6-O-[2-deoxy-3-O-(3-metoxydecyl)-6-methyl-2-[(1-oxo-11-octadecenyl)amino]-4-O-phosphono-β-D-glucopyranosyl]-2-[(1,3-dioxotetradecyl)amino]-α-D-glucopyranose 1-(dihydrogen phosphate) tetrasodium salt

2932 99 00

136172-58-2

1,6-di-O-acetyl-2-azido-3,4-di-O-benzyl-2-deoxy-D-glucopyranose

2932 99 00

196597-80-5

2-[(8S)-1,6,7,8-tetrahydro-2H-indeno[5,4-b]furan-8-yl]ethanamine hydrochloride

2932 99 00

666860-59-9

2-amino-2-oxoethyl{3-[trans-5-(6-methoxynaphthalen-1-yl)-1,3-dioxan-2-yl]propyl}carbamate

2932 99 00

117661-72-0

5-(chloromethyl)-6-methyl-1,3-benzodioxole

2932 99 00

959624-24-9

6-(hydroxymethyl)-4-phenyl-3,4-dihydro-2H-chromen-2-ol

2932 99 00

960404-59-5

but-2-yne-1,4-diol – methyl 1-C-[4-chloro-3-(4-ethoxybenzyl)phenyl]-α-D-glucopyranoside (1:1)

2932 99 00

15826-37-6

disodium 5,5′-[(2-hydroxypropane-1,3-diyl)bis(oxy)]bis(4-oxo-4H-chromene-2-carboxylate)

2932 99 00

204254-84-2

ethyl (3aR,7R,7aR)-2,2-dimethyl-7-[(methylsulfonyl)oxy]-3a,6,7,7a-tetrahydro-1,3-benzodioxole-5-carboxylate

2932 99 00

99541-26-1

methyl (2S,3S,4S,5S,6S)-6-{[(1S,2S,3S,4R,5R)-3-(acetyloxy)-4-azido-6,8-dioxabicyclo[3.2.1]oct-2-yl]methyl}-4,5-bis(benzyloxy)-3-hydroxytetrahydro-2H-pyran-2-carboxylate

2932 99 00

114869-97-5

methyl 6-O-acetyl-4-O-(2-O-acetyl-3-O-benzyl-6-methyl-α-L-idopyranuronosyl)-3-O-benzyl-2-{[(benzyloxy)carbonyl]amino}-2-deoxy-α-D-glucopyranoside

2933 19 90

1035677-60-1

(4S)-3-(4-chlorophenyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide 2,3-dihydroxybutanedioate

2933 19 90

18048-64-1

2-(3,4-dimethylphenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one

2933 19 90

1035675-24-1

3-(4-chlorophenyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide

2933 19 90

1028026-83-6

5-methyl-1-(propan-2-yl)-4-[4-(propan-2-yloxy)benzyl]-1,2-dihydro-3H-pyrazol-3-one

2933 19 90

473921-12-9

5-{[3,5-diethyl-1-(2-hydroxyethyl)-1H-pyrazol-4-yl]oxy}benzene-1,3-dicarbonitrile

2933 29 90

65902-59-2

2-bromo-4-nitro-1H-imidazole

2933 29 90

57531-37-0

2-chloro-4-nitro-1H-imidazole

2933 29 90

1000164-35-1

3-(1,1-dimethylethyl)-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-1-(triphenylmethyl)-L-histidyl-2-methylalanyl-L-α-glutamylglycine

2933 29 90

152074-97-0

L-α-aspartyl-L-α-glutamyl-L-asparaginyl-L-prolyl-L-valyl-L-valyl-L-histidyl-L-phenylalanyl-L-phenylalanyl-L-lysyl-L-asparaginyl-L-isoleucyl-L-valyl-L-threonyl-L-prolyl-L-arginyl-L-threonine

2933 29 90

781666-30-6

L-α-aspartyl-L-α-glutamyl-L-asparaginyl-L-prolyl-L-valyl-L-valyl-L-histidyl-L-phenylalanyl-L-phenylalanyl-L-lysyl-L-asparaginyl-L-isoleucyl-L-valyl-L-threonyl-L-prolyl-L-arginyl-L-threonine tetraacetate

2933 29 90

451470-33-0

methyl 3′-(2-methyl-4,5-dihydro-1H-imidazol-1-yl)biphenyl-3-carboxylate

2933 39 99

925978-49-0

(+)-5-[6-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl]-1-azabicyclo[3.2.1]octane

2933 39 99

876170-44-4

(1S,5S)-3-(5,6-dichloropyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane benzenesulfonate

2933 39 99

741705-70-4

(2R)-phenyl[(2R)-piperidin-2-yl]ethanoic acid hydrochloride

2933 39 99

414910-13-7

(2S)-hydroxy(phenyl)ethanoic acid – (2R)-2-(4-fluoro-2-methylphenyl)piperidin-4-one (1:1)

2933 39 99

0-00-0

(3aR,6aR)-1-(pyridin-3-yl)octahydropyrrolo[3,4-b]pyrrole 4-methylbenzenesulfonate

2933 39 99

370882-57-8

(3aR,6aR)-1-(pyridin-3-yl)octahydropyrrolo[3,4-b]pyrrole dihydrochloride

2933 39 99

334618-23-4

(3R)-piperidin-3-amine dihydrochloride

2933 39 99

1062580-52-2

(3R,4R)-1-benzyl-N,4-dimethylpiperidin-3-amine dihydrochloride

2933 39 99

27262-47-1

(S)-1-butyl-N-(2,6-dimethylphenyl)piperidine-2-carboxamide

2933 39 99

105812-81-5

[(3S,4R)-4-(4-fluorophenyl)-1-methylpiperidin-3-yl]methanol

2933 39 99

876068-51-8

[(3S,4S)-4-amino-1-(5,6-dichloropyridin-3-yl)pyrrolidin-3-yl]methanol

2933 39 99

871022-14-9

1-({4-[({[2-oxo-3-(propan-2-yl)-2,3-dihydro-1H-benzimidazol-1-yl]carbonyl}amino)methyl]piperidin-1-yl}methyl)cyclobutanecarboxylic acid

2933 39 99

5421-92-1

1-(pyridin-4-yl)pyridinium chloride hydrochloride

2933 39 99

272776-12-2

1,1′-binaphthalene-2,2′-diol –5-methoxy-2-{(S)-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfinyl}-1H-benzimidazole (1:1)

2933 39 99

871022-19-4

1-[(4-{[(tert-butoxycarbonyl)amino]methyl}piperidin-1-yl)methyl]cyclobutanecarboxylic acid

2933 39 99

3613-73-8

2,8-dimethyl-5-[2-(6-methylpyridin-3-yl)ethyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole

2933 39 99

179687-79-7

2-[(2-chloro-4-nitrophenoxy)methyl]pyridine

2933 39 99

122321-04-4

2-[methyl(pyridin-2-yl)amino]ethanol

2933 39 99

945405-37-8

2-methyl-3-[(2S)-pyrrolidin-2-ylmethoxy]pyridine 2,3-dihydroxybutanedioate

2933 39 99

936637-40-0

3,3′-piperidine-1,4-diyldipropan-1-ol 4-methylbenzenesulfonate

2933 39 99

88150-62-3

3-ethyl-5-methyl-4-(2-chlorophenyl)-2-{[2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethoxy]methyl}-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate

2933 39 99

84100-54-9

4-(ethylamino)piperidine-4-carboxamide

2933 39 99

873546-30-6

4,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]bis(N′-hydroxybenzenecarboximidamide)

2933 39 99

873546-74-8

4,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]bis[N′-(acetyloxy)benzenecarboximidamide]

2933 39 99

873546-38-4

4,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]dibenzenecarboximidamide trihydrochloride pentahydrate

2933 39 99

873546-80-6

4,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]dibenzonitrile

2933 39 99

78750-61-5

4-[(3-nitropyridin-2-yl)amino]phenol

2933 39 99

866109-93-5

4-{4-[4-(trifluoromethoxy)phenoxy]piperidin-1-yl}phenol 4-methylbenzenesulfonate

2933 39 99

927889-51-8

4-bromo-2,6-diethylpyridine 4-methylbenzenesulfonate

2933 39 99

691882-47-0

4-hydroxybenzoic acid – (2S,4E)-N-methyl-5-[5-(propan-2-yloxy)pyridin-3-yl]pent-4-en-2-amine (1:1)

2933 39 99

876068-46-1

5,6-dichloro-N-(2,2-dimethoxyethyl)pyridin-3-amine

2933 39 99

1072-98-6

5-chloropyridin-2-amine

2933 39 99

298692-34-9

6-(chloroacetyl)pyridine-2-carboxylic acid

2933 39 99

550349-58-1

7-chloro-3-(6-methoxypyridin-3-yl)-N,N,5-trimethyl-4-oxo-4,5-dihydro-3H-pyridazino[4,5-b]indole-1-carboxamide

2933 39 99

414909-98-1

benzyl 2-(4-fluoro-2-methylphenyl)-4-oxo-3,4-dihydropyridine-1(2H)-carboxylate

2933 39 99

56880-11-6

ethyl [(3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl)acetate

2933 39 99

548797-97-3

N-(2-{[(2S)-3-{[1-(4-chlorobenzyl)piperidin-4-yl]amino}-2-hydroxy-2-methylpropyl]oxy}-4-hydroxyphenyl)acetamide

2933 39 99

0-00-0

N-[(S)-1-azabicyclo[2.2.2]oct-2-yl(phenyl)methyl]-2,6-dichloro-3-(trifluoromethyl)benzamide hydrochloride

2933 39 99

329003-65-8

sodium hydrogen [1-hydroxy-1-phosphono-2-(pyridin-3-yl)ethyl]phosphonate hemipentahydrate

2933 49 10

417716-92-8

4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide methanesulfonate

2933 49 90

503291-53-0

2-ethylbutyl (3S,4aS,6S,8aR)-6-[3-chloro-2-(1H-tetrazol-5-yl)phenoxy]decahydro-3-isoquinolinecarboxylate 4-methylbenzenesulfonate

2933 49 90

103733-32-0

benzyl (3S)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylate hydrochloride

2933 49 90

503293-98-9

(3S,4aS,6S,8aR)-6-hydroxy-2-(methoxycarbonyl)decahydroisoquinoline-3-carboxylic acid

2933 49 90

503290-66-2

(3S,4aS,6S,8aR)-6-[3-chloro-2-(2H-tetrazol-5-yl)phenoxy]decahydro-3-isoquinolinecarboxylic acid hydrochloride

2933 49 90

134388-95-7

(3S,4aS,8aR)-2-(methoxycarbonyl)-6-oxodecahydroisoquinoline-3-carboxylic acid – (1R)-1-phenylethanamine (1:1)

2933 49 90

868210-14-4

4-(4-{[(2S,4R)-4-[acetyl(4-chlorophenyl)amino]-2-methyl-3,4-dihydroquinolin-1(2H)-yl]carbonyl}phenoxy)-2,2-dimethylbutanoic acid

2933 49 90

00-00-0

methyl 2-[(3R)-3-{3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl}-3-({[1-(hydroxymethyl)cyclopropyl]methyl}sulfanyl)propyl]benzoate hydrochloride

2933 49 90

848133-76-6

N-(4-chloro-3-cyano-7-ethoxyquinolin-6-yl)acetamide

2933 59 95

869490-23-3

(3,3-difluoropyrrolidin-1-yl){(2S,4S)-4-[4-(pyrimidin-2-yl)piperazin-1-yl]pyrrolidin-2-yl}methanone

2933 59 95

941685-40-1

(3R)-3-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile

2933 59 95

941678-49-5

(3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile

2933 59 95

941685-41-2

(3S)-3-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile

2933 59 95

957187-34-7

[(8R)-8-(3,5-difluorophenyl)-10-oxo-6,9-diazaspiro[4.5]dec-9-yl]acetic acid

2933 59 95

356058-42-9

{2-[(4-fluorobenzyl)sulfanyl]-4-oxo-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidin-1-yl}acetic acid

2933 59 95

0-00-0

2,3-dihydroxy-2,3-bis(phenylcarbonyl)butanedioic acid – ethyl [(8R)-8-(3,5-difluorophenyl)-10-oxo-6,9-diazaspiro[4.5]dec-9-yl]acetate (1:1)

2933 59 95

90213-66-4

2,4-dichloro-7H-pyrrolo[2,3-d]pyrimidine

2933 59 95

3934-20-1

2,4-dichloropyrimidine

2933 59 95

451487-18-6

2-[(4-fluorobenzyl)sulfanyl]-1,5,6,7-tetrahydro-4H-cyclopenta[d]pyrimidin-4-one

2933 59 95

865758-96-9

2-[(6-chloro-3-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methyl]benzonitrile

2933 59 95

934815-71-1

2-[3-(6-{[2-(2,4-dichlorophenyl)ethyl]amino}-2-methoxypyrimidin-4-yl)phenyl]-2-methylpropanoic acid phosphate

2933 59 95

722543-31-9

2-{ethyl[3-({4-[(5-{2-[(3-fluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]quinazolin-7-yl}oxy)propyl]amino}ethyl dihydrogen phosphate

2933 59 95

1032066-96-8

2-amino-9-{(1S,3R,4S)-3-[(benzyloxy)methyl]-4-[dimethyl(phenyl)silyl]-2-methylidenecyclopentyl}-1,9-dihydro-6H-purin-6-one – methanesulfonate (2:1)

2933 59 95

540737-29-9

3-{(3R,4R)-4-methyl-3-[methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile 2-hydroxypropane-1,2,3-tricarboxylate

2933 59 95

1137917-12-4

3-{[6-(ethylsulfonyl)pyridin-3-yl]oxy}-5-{[(2S)-1-hydroxypropan-2-yl]oxy}benzoic acid – 1,4-diazabicyclo[2.2.2]octane (2:1)

2933 59 95

941685-39-8

3-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile

2933 59 95

941685-27-4

4-(1H-pyrazol-4-yl)-7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidine

2933 59 95

1780-26-3

4,6-dichloro-2-methylpyrimidine

2933 59 95

145783-14-8

4,6-dichloro-5-nitro-2-(propylsulfanyl)pyrimidine

2933 59 95

3680-69-1

4-chloro-7H-pyrrolo[2,3-d]pyrimidine

2933 59 95

61379-64-4

4-cyclopentylpiperazin-1-amine

2933 59 95

55112-42-0

4-methylpiperazine-1-carbonyl chloride hydrochloride

2933 59 95

0-00-0

5-(benzylamino)-2-(3-methoxyphenyl)-7-(4-methylpiperazin-1-yl)[1,2,4]triazolo[1,5-a]quinoline-4-carbonitrile – (2E)-but-2-enedioate (2:1) hydrate

2933 59 95

55293-96-4

5,7-dimethyl[1,2,4]triazolo[1,5-a]pyrimidine-2-carbaldehyde

2933 59 95

179688-01-8

7-(benzyloxy)-6-methoxyquinazolin-4(3H)-one

2933 59 95

444731-74-2

N-(2-chloropyrimidin-4-yl)-2,3-dimethyl-2H-indazol-6-amine

2933 59 95

0-00-0

N-(5-fluoro-3-methyl-1H-indol-1-yl)-4-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide

2933 79 00

586414-48-4

(-)-3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2H)-yl}-N,4-dimethylbenzamide

2933 79 00

425663-71-4

(1S)-1-amino-3-methyl-1,3,4,5-tetrahydro-2H-3-benzazepin-2-one hydrochloride

2933 79 00

813452-14-1

(4S)-1-[(2S,3S,11bS)-2-amino-9,10-dimethoxy-1,3,4,6,7,11b-hexahydro-2H-pyrido[2,1-a]isoquinolin-3-yl]-4-(fluoromethyl)pyrrolidin-2-one dihydrochloride

2933 79 00

5162-90-3

3-(2-oxo-1,2-dihydroquinolin-4-yl)alanine

2933 79 00

536760-29-9

3-chloro-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one

2933 79 00

4876-10-2

4-(bromomethyl)quinolin-2(1H)-one

2933 79 00

5057-12-5

4,6,7,8-tetrahydroquinoline-2,5(1H,3H)-dione

2933 79 00

54197-66-9

6-hydroxy-3,4-dihydroquinolin-2(1H)-one

2933 79 00

22246-18-0

7-hydroxy-3,4-dihydroquinolin-2(1H)-one

2933 79 00

536759-91-8

ethyl 1-(4-methoxyphenyl)-6-(4-nitrophenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate

2933 79 00

503614-91-3

ethyl 1-(4-methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate

2933 79 00

586379-61-5

methyl 3-(4-hydroxy-6-methyl-2-oxopyridin-1(2H)-yl)-4-methylbenzoate

2933 99 80

709031-45-8

(1S,3S,5S)-2-azabicyclo[3.1.0]hexane-3-carboxamide methanesulfonate

2933 99 80

649735-46-6

(2R)-1-({4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl}oxy)propan-2-ol

2933 99 80

51077-14-6

(2S)-1-(tert-butoxycarbonyl)azetidine-2-carboxylic acid

2933 99 80

631916-97-7

(2S)-N-{4-[(Z)-amino(methoxyimino)methyl]benzyl}-1-{(2R)-2-[3-chloro-5-(difluoromethoxy)phenyl]-2-hydroxyethanoyl}azetidine-2-carboxamide – benzenesulphonic acid (1:1)

2933 99 80

80875-98-5

(2S,3aS,7aS)-octahydro-1H-indole-2-carboxylic acid

2933 99 80

948846-40-0

(2S,3S)-2,3-bis[(phenylcarbonyl)oxy]butanedioic acid – ethyl (3aR,6aR)-hexahydropyrrolo[3,4-b]pyrrole-5(1H)-carboxylate (1:1)

2933 99 80

1000164-36-2

(5S,8S,11S,14S,17S,20S,23S,26S,29S,32S,35S,38S)-5-(3-amino-3-oxopropyl)-20-benzyl-23-[(2S)-butan-2-yl]-14,38-bis{4-[(tert-butoxycarbonyl)amino]butyl}-29-{[1-(tert-butoxycarbonyl)-1H-indol-3-yl]methyl}-17-(3-tert-butoxy-3-oxopropyl)-1-(1H-fluoren-9-yl)-8,11,26,41,41-pentamethyl-32-(2-methylpropyl)-3,6,9,12,15,18,21,24,27,30,33,36,39-tridecaoxo-35-(propan-2-yl)-2-oxa-4,7,10,13,16,19,22,25,28,31,34,37,40-tridecaazadotetracontan-42-oic acid

2933 99 80

22162-51-2

1-(2-nitrobenzyl)-1H-pyrrole-2-carbaldehyde

2933 99 80

35681-40-4

1-(propan-2-yl)-1,3-dihydro-2H-benzimidazol-2-one

2933 99 80

166170-15-6

1-(tert-butoxycarbonyl)-2-methyl-D-proline

2933 99 80

796967-16-3

1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-5-methylphenyl)urea

2933 99 80

0-00-0

1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-5-methylphenyl)urea hydrochloride

2933 99 80

444731-72-0

2,3-dimethyl-2H-indazol-6-amine

2933 99 80

19686-05-6

2,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole

2933 99 80

912444-00-9

2-[(2R)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide

2933 99 80

912445-36-4

2-[(2S)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide dihydrochloride

2933 99 80

163457-23-6

3,3-difluoropyrrolidine hydrochloride

2933 99 80

239463-85-5

3-{5-[(2R)-2-aminopropyl]-7-cyano-2,3-dihydro-1H-indol-1-yl}propyl benzoate (2R,3R)-2,3-dihydroxybutanedioate

2933 99 80

55321-99-8

3-oxo-3,4-dihydropyrazine-2-carboxamide

2933 99 80

952490-01-6

4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl 2,2-dimethylpropanoate

2933 99 80

942436-93-3

4-amino-8-(2,5-dimethoxyphenyl)-N-propylcinnoline-3-carboxamide

2933 99 80

942437-37-8

4-amino-8-(2-fluoro-6-methoxyphenyl)-N-propylcinnoline-3-carboxamide

2933 99 80

288385-88-6

4-fluoro-2-methyl-1H-indol-5-ol

2933 99 80

503293-47-8

5-(2-chloro-6-fluorophenyl)-2H-tetrazole

2933 99 80

73963-42-5

5-(4-chlorobutyl)-1-cyclohexyl-1H-tetrazole

2933 99 80

606143-52-6

5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-N-(2-hydroxyethoxy)-1-methyl-1H-benzimidazole-6-carboxamide

2933 99 80

0-00-0

5-fluoro-1-(3-fluorobenzyl)-N-(1H-indol-5-yl)-1H-indole-2-carboxamide

2933 99 80

872206-47-8

5-methyl-4-oxo-1,4-dihydropyrrolo[2,1-f][1,2,4]triazin-6-yl 2,2-dimethylpropanoate

2933 99 80

259793-88-9

6-bromo-3-oxo-3,4-dihydropyrazine-2-carboxamide

2933 99 80

1137606-74-6

6-fluoro-3-oxo-3,4-dihydropyrazine-2-carbonitrile – N-cyclohexylcyclohexanamine (1:1)

2933 99 80

261953-36-0

6-iodo-1H-indazole

2933 99 80

80076-47-7

8,9-difluoro-5-methyl-1-oxo-6,7-dihydro-1H,5H-pyrido[3,2,1-ij]quinoline-2-carboxylic acid

2933 99 80

52602-39-8

9H-carbazol-4-ol

2933 99 80

145641-35-6

benzyl (2S,3aR,7aS)-octahydro-1H-indole-2-carboxylate hydrochloride

2933 99 80

87269-87-2

benzyl (2S,3aS,6aS)-octahydrocyclopenta[b]pyrrole-2-carboxylate hydrochloride

2933 99 80

1012065-72-3

ethyl 2-amino-9,10-dimethoxy-1,6,7,11b-tetrahydro-4H-pyrido[2,1-a]isoquinoline-3-carboxylate

2933 99 80

131707-24-9

ethyl 6-bromo-5-hydroxy-1-methyl-2-[(phenylsulfanyl)methyl]-1H-indole-3-carboxylate

2933 99 80

105152-95-2

ethyl 7-(3-aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylate

2933 99 80

139481-44-0

methyl 1-[(2′-cyanobiphenyl-4-yl)methyl]-2-ethoxy-1H-benzimidazole-7-carboxylate

2933 99 80

0-00-0

methyl 1-tert-butyl-2-hydroxy-1H-pyrrolo[2,3-b]pyridine-3-carboxylate

2933 99 80

21688-11-9

N2-[(benzyloxy)carbonyl]-L-glutaminyl-L-asparaginyl-S-benzyl-L-cysteinyl-L-prolyl-L-leucylglycinamide

2933 99 80

361440-67-7

tert-butyl (1S,3S,5S)-3-carbamoyl-2-azabicyclo[3.1.0]hexane-2-carboxylate

2933 99 80

709031-38-9

tert-butyl (2S)-2-carbamoyl-2,3-dihydro-1H-pyrrole-1-carboxylate

2933 99 80

709031-43-6

tert-butyl [(1S)-2-[(1S,3S,5S)-3-cyano-2-azabicyclo[3.1.0]hex-2-yl]-1-(3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl)-2-oxoethyl]carbamate

2933 49 90

936359-25-0

methyl 2-((R)-3-(3-((E)-2-(7-chloroquinolin-2-yl)vinyl)phenyl)-3-(((1-(hydroxymethyl)cyclopropyl)methyl)sulfanyl)propyl)benzoate

2934 10 00

110130-88-6

(2Z)-[(acetyloxy)imino](2-amino-1,3-thiazol-4-yl)ethanoic acid

2934 10 00

68672-66-2

(2Z)-{[(1-tert-butoxy-2-methyl-1-oxopropan-2-yl)oxy]imino}[2-(tritylamino)-1,3-thiazol-4-yl]ethanoic acid

2934 10 00

291536-35-1

(5Z)-5-(4-fluorobenzylidene)-1,3-thiazolidine-2,4-dione

2934 10 00

302964-24-5

2-amino-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide

2934 10 00

866920-24-3

3-[2-chloro-4-({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methoxy)phenyl]-1,2,4-oxadiazol-5(4H)-one

2934 10 00

752253-39-7

4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(prop-2-yn-1-yl)-1,3-thiazol-2-amine

2934 10 00

914361-45-8

L-lysine – {[(2R,3R)-3-[4-(4-cyanophenyl)-1,3-thiazol-2-yl]-2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butan-2-yl]oxy}methyl dihydrogen phosphate – ethanol (1:1:1)

2934 10 00

302964-08-5

N-(2-chloro-6-methylphenyl)-2-[(6-chloro-2-methylpyrimidin-4-yl)amino]-1,3-thiazole-5-carboxamide

2934 10 00

127660-04-2

sodium (2Z)-(2-amino-1,3-thiazol-4-yl)(hydroxyimino)ethanoate

2934 99 90

17381-54-3

(1-benzothiophen-5-yl)acetic acid

2934 99 90

630100-90-2

(1R)-1,2-anhydro-4-C-{(1E,3E)-4-[(1S,2S,3E,5R,6R,9R)-5-(1-carboxylato-4-cycloheptylpiperazin-2-yl)-6,9-dihydroxy-2,6-dimethyl-11-oxooxacyclododec-3-en-1-yl]penta-1,3-dien-1-yl}-3,5-dideoxy-1-[(2R,3S)-3-hydroxypentan-2-yl]-D-erythropentitol

2934 99 90

220099-91-2

(2R)-3′H-spiro[4-azabicyclo[2.2.2]octane-2,2′-furo[2,3-b]pyridine]

2934 99 90

220100-81-2

(2R)-3′H-spiro[4-azabicyclo[2.2.2]octane-2,2′-furo[2,3-b]pyridine] (S,S)-2,3-dihydroxybutanedioate

2934 99 90

161599-46-8

(2R,3R,4R,5R)-2-(4-amino-5-fluoro-2-oxopyrimidin-1(2H)-yl)-2-fluoro-5-methyltetrahydrofuran-3,4-diyl diacetate

2934 99 90

690270-65-6

(2R,3S,4R)-5-(4-amino-2-oxopyrimidin-1(2H)-yl)-2-azido-2-{[(2-methylpropanoyl)oxy]methyl}tetrahydrofuran-3,4-diyl bis(2-methylpropanoate) hydrochloride

2934 99 90

265121-04-8

(3-{[(2R,3S)-2-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy}-3-(2-fluorophenyl)morpholin-4-yl]methyl}-5-oxo-2,5-dihydro-1H-1,2,4-triazol-1-yl)phosphonic acid – 1-deoxy-1-(methylamino)-D-glucitol (1:2)

2934 99 90

163680-80-6

(3S)-10-[1-(acetylamino)cyclopropyl]-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7H-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxylic acid

2934 99 90

132335-46-7

(3S)-N,N-dimethyl-3-(naphthalen-1-yloxy)-3-(thiophen-2-yl)propan-1-amine

2934 99 90

133413-70-4

(3S,6R,9S,12R,15S,18R,21S,24R)-6,18-dibenzyl-4,10,12,16,22,24-hexamethyl-3,9,15,21-tetrakis(2-methylpropyl)-1,7,13,19-tetraoxa-4,10,16,22-tetraazacyclotetracosane-2,5,8,11,14,17,20,23-octone

2934 99 90

503068-36-8

(5R)-3-(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl)-5-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-1,3-oxazolidin-2-one

2934 99 90

452339-73-0

(5R)-5-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-1,3-oxazolidin-2-one

2934 99 90

877130-28-4

(6R)-6-cyclopentyl-6-[2-(2,6-diethylpyridin-4-yl)ethyl]-3-[(5,7-dimethyl[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methyl]-4-hydroxy-5,6-dihydro-2H-pyran-2-one

2934 99 90

132335-44-5

(S)-3-(dimethylamino)-1-(thiophen-2-yl)propan-1-ol

2934 99 90

812647-80-6

{(2R,3S,4R,5R)-2-azido-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-bis[(phenylcarbonyl)oxy]tetrahydrofuran-2-yl}methyl 3-chlorobenzoate

2934 99 90

00-00-0

1-(1-{4-[2-(4-fluorophenyl)-1,3-dioxolan-2-yl]butyl}-1,2,3,6-tetrahydropyridin-4-yl)-1,3-dihydro-2H-benzimidazol-2-one

2934 99 90

1029716-44-6

1-(1-ethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole

2934 99 90

165172-60-1

1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]-5-methylpyrimidine-2,4(1H,3H)-dione – 1-methylpyrrolidin-2-one (1:1)

2934 99 90

519187-97-4

1-[3-(2-benzo[b]thien-5-ylethoxy)propyl]-3-azetidinol – (2Z)-2-butenedioate (1:1)

2934 99 90

127000-90-2

1-{[(2R,3S)-2-(2,4-difluorophenyl)-3-methyloxiran-2-yl]methyl}-1H-1,2,4-triazole

2934 99 90

710281-33-7

2-({[(1R,3S)-3-{[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}cyclohexyl]oxy}methyl)-6-methylbenzoic acid

2934 99 90

96803-30-4

2-(1-benzothiophen-5-yl)ethanol

2934 99 90

913695-00-8

2-[({4-[(2,2-dimethyl-1,3-dioxan-5-yl)methoxy]-3,5-dimethylpyridin-2-yl}methyl)sulfinyl]-1Hbenzimidazole, sodium salt (1:1)

2934 99 90

376608-74-1

2-{[(3aR,4S,6R,6aS)-6-{[5-amino-6-chloro-2-(propylsulfanyl)pyrimidin-4-yl]amino}-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl]oxy}ethanol

2934 99 90

474554-48-8

2-bromo-1-[3-tert-butyl-4-methoxy-5-(morpholin-4-yl)phenyl]ethanone

2934 99 90

530141-72-1

3-(5-{[4-(cyclopentyloxy)-2-hydroxyphenyl]carbonyl}-2-[(3-hydroxy-1,2-benzoxazol-6-yl)methoxy]phenyl)propanoic acid

2934 99 90

519188-55-7

3-[2-(1-benzothiophen-5-yl)ethoxy]-1-(3-hydroxyazetidin-1-yl)propan-1-one

2934 99 90

519188-42-2

3-[2-(1-benzothiophen-5-yl)ethoxy]propionic acid

2934 99 90

753015-42-8

3-{(E)-2-[(3R)-pyrrolidin-3-yl]ethenyl}-5-(tetrahydro-2H-pyran-4-yloxy)pyridine

2934 99 90

26638-53-9

3-chloro-6-methyldibenzo[c,f][1,2]thiazepin-11(6H)-one 5,5-dioxide

2934 99 90

499785-81-8

3-oxo-4-(2,3,5-tri-O-acetyl-β-D-ribofuranosyl)-3,4-dihydropyrazine-2-carboxamide

2934 99 90

356782-84-8

3-oxo-4-(β-D-ribofuranosyl)-3,4-dihydropyrazine-2-carboxamide

2934 99 90

6504-57-0

4-[3-hydroxy-3-phenyl-3-(thiophen-2-yl)propyl]-4-methylmorpholin-4-ium methyl sulfate

2934 99 90

871484-32-1

4-[4-({3-[(4-deoxy-4-fluoro-b-D-glucopyranosyl)oxy]-5-(propan-2-yl)-1H-pyrazol-4-yl}methyl)phenyl]-N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]butanamide

2934 99 90

166964-09-6

4-chloro-3-methyl-1,2-oxazol-5-amine

2934 99 90

655233-39-3

4-nitrobenzyl(6R,7R)-7-amino-8-oxo-3-[(2S)-tetrahydrofuran-2-yl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate hydrochloride

2920 90 85

89729-09-9

5,7-dioxa-6-thiaspiro[2.5]octane-6-oxide

2934 99 90

388082-75-5

5-[4-[[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]amino]-6-quinazolinyl]-2-furancarboxaldehyde – 4-methylbenzenesulfonate (1:1)

2934 99 90

4923-87-9

5-bromo-1-benzothiophene

2934 99 90

947408-95-9

6-(bromomethyl)-2-triphenylmethyl-1,2-benzisoxazol-3(2H)-one

2934 99 90

947408-94-8

6-methyl-2-trityl-1,2-benzoxazol-3(2H)-one

2934 99 90

67978-05-6

diphenylmethyl(2R)-3-methyl-2-[(1R,5S)-3-(4-methylphenyl)-7-oxo-4-oxa-2,6-diazabicyclo[3.2.0]hept-2-en-6-yl]but-3-enoate

2934 99 90

1001859-46-6

DNA (synthetic plasmid vector pCOR human interferon beta signal peptide fusion protein with 21-154-human acidic fibroblast growth factor-specifying)

2934 99 90

665058-78-6

DNA, d(T-sp-C-G-sp-T-sp-C-G-sp-T-sp-T-sp-T-sp-T-sp-G-sp-A-sp-C-G-sp-T-sp-T-sp-T-sp-T-sp-Gsp-T-sp-C-G-sp-T-sp-T)

2934 99 90

923591-06-4

methyl (5R,7S,10S)-10-tert-butyl-15,15-dimethyl-3,9,12-trioxo-6,7,9,10,11,12,14,15,16,17,18,19-dodecahydro-1H,5H-2,23:5,8-dimethano-4,13,2,8,11-benzodioxatriazacyclohenicosine-7(3H)-carboxylate

2934 99 90

59337-92-7

methyl 3-(chlorosulfonyl)thiophene-2-carboxylate

2934 99 90

947409-01-0

methyl 3-[5-[4-(cyclopentyloxy)-2-hydroxybenzoyl]-2-[(2-triphenylmethyl-1,2-benzisoxazol-3(2H)-on-6-yl)methoxy]phenyl]propionate

2934 99 90

85006-31-1

methyl 3-amino-4-methylthiophene-2-carboxylate

2934 99 90

893428-72-3

N-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methyl-1-piperazinyl)ethoxy]-5-[(tetrahydro-2H-pyran-4-yl)oxy]-4-quinazolinamine – (2E)-2-butenedioate (1:2)

2934 99 90

390800-88-1

N,N′,N′′-(boroxin-2,4,6-triyltris{[(1S)-3-methylbutane-1,1-diyl]imino[(2S)-1-oxo-3-phenylpropane-1,2-diyl]})tripyrazine-2-carboxamide

2934 99 90

112913-94-7

N-{[4-(4-fluorobenzyl)morpholin-2-yl]methyl}acetamide

2934 99 90

120788-03-6

S-[(1R,3S)-1-oxidotetrahydrothiophen-3-yl] ethanethioate

2935 00 90

1198178-65-2

(1R,2R)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethylcyclopropanaminium 4-methylbenzenesulfonate

2935 00 90

39570-96-2

(2R)-3-(benzylsulfanyl)-N-[(2S)-1-{[(2S,3S)-1-hydrazinyl-3-methyl-1-oxopentan-2-yl]amino}-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-2-{[(4-methylphenyl)sulfonyl]amino}propanamide

2935 00 90

24310-36-9

1-[(4-methylphenyl)sulfonyl]-1,2,3,4-tetrahydro-5H-1-benzazepin-5-one

2935 00 90

0-00-0

2-(cyclohexylmethyl)-N-{2-[(2S)-1-methylpyrrolidin-2-yl]ethyl}-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide di[(2E)-but-2-enedioate] hydrate

2935 00 90

941690-55-7

3-[(methylsulfonyl)amino]-2-phenyl-N-[(1S)-1-phenylpropyl]quinoline-4-carboxamide

2935 00 90

6973-09-7

5-amino-2-methylbenzenesulfonamide

2935 00 90

193686-76-9

7-chloro-1-[(4-methylphenyl)sulfonyl]-1,2,3,4-tetrahydro-5H-1-benzazepin-5-one

2935 00 90

123664-84-6

N-(5-methoxy-2-phenoxyphenyl)methanesulfonamide

2935 00 90

149457-03-4

N-[4-(N-formylglycyl)-5-hydroxy-2-phenoxyphenyl]methanesulfonamide

2935 00 90

149456-98-4

N-[4-(N-formylglycyl)-5-methoxy-2-phenoxyphenyl]methanesulfonamide

2935 00 90

141450-48-8

N-{2-[(4-hydroxyphenyl)amino]pyridin-3-yl}-4-methoxybenzenesulfonamide hydrochloride

2935 00 90

289042-10-0

N-{5-[(diphenylphosphoryl)methyl]-4-(4-fluorophenyl)-6-(propan-2-yl)pyrimidin-2-yl}-N-methylmethanesulfonamide

2939 99 00

7689-03-4

(4S)-4-ethyl-4-hydroxy-1H-pyrano[3′,4′:6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione

2939 99 00

477-29-2

colchicoside

2940 00 00

604-69-3

1,2,3,4,6-penta-O-acetyl-β-D-glucopyranose

2940 00 00

647834-15-9

2-(4-methoxybenzyl)thiophen-3-yl β-D-glucopyranoside

2941 90 00

76610-92-9

(6R,7R)-7-({N-[(4-ethyl-2,3-dioxopiperazin-1-yl)carbonyl]-D-threonyl}amino)-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid

3907 20 99

913976-27-9

poly(oxy-1,2-ethanediyl), α-hydro-ω-methoxy, diester with 21N6, 21′N6-[[(N2, N6-dicarboxy-L-lysyl-β-alanyl)imino]bis(1-oxo-2, 1-ethanediyl)]bis[N-acetylglycyl-L-leucyl-L-tyrosyl-L-alanyl-L-cysteinyl-L-histidyl-L-methionylglycyl-L-prolyl-L-isoleucyl-L-threonyl-3-(1-naphthalenyl)-L-alanyl-L-valyl-L-cysteinyl-L-glutaminyl-L-prolyl-L-leucyl-L-arginyl-N-methylglycyl-L-lysinamide] cyclic (6→15), (6′→15′) bis(disulfide)


ANNEX IV

List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be withdrawn from the list of products receiving duty-free treatment included in Annex 6 to Annex I to Regulation (EEC) No 2658/87 due to their transfer to the list of products receiving duty-free treatment included in Annex 3 to Annex I to Regulation (EEC) No 2658/87

CN code

CAS RN

Name

2915 39 00

2937 29 00

7753-60-8

17-alpha-hydroxy-3,20-dioxopregna-4,9(11)-diene-21-yl acetate

see anecortave (INN)

2920 90 85

163133-43-5

4-(nitrooxy)butyl (2S)-2-(6-methoxy-2-naphthyl) propanoate

see naproxcinod (INN)

2924 29 98

194085-75-1

2-(2-chlorophenyl)-2-hydroxyethyl carbamate

see carisbamate (INN)

2933 39 99

103129-82-4

3-ethyl 5-methyl 2-[(2-aminoethoxy)methyl]-4-(2-chlorophenyl)-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate

see levamlodipine (INN)

2933 39 99

319460-85-0

N-methyl-2-{[3-((E)-2-pyridin-2-ylvinyl)-1H-indazol-6-yl]sulfanyl}benzamide

see axitinib (INN)

2934 10 00

302962-49-8

N-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)thiazole-5-carboxamide

see dasatinib (INN)

2934 99 90

143491-57-0

(2R,5S)-4-amino-5-fluoro-1-[2-(hydroxymethyl)-1,3-oxathiolan-5-yl]pyrimidin-2(1H)-one

see emtricitabine(INN)

2934 99 90

98819-76-2

(2S)-2-[(S)-(2-ethoxyphenoxy)phenylmethyl]morpholine

see esreboxetine (INN)

2934 99 90

475479-34-6

(2S)-2-methoxy-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]-1-benzothiophen-7-yl}propanoic acid

see aleglitazar (INN)

2934 99 90

377727-87-2

2-(2-furyl)-7-(2-{4-[4-(2-methoxyethoxy)phenyl] piperazin-1-yl}ethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[2,3-c]pyrimidin-5-amine

see preladenant (INN)

2934 99 90

189003-92-7

2-{7-fluoro-2-oxo-4-[2-(4-thieno[3,2-c]pyridin-4-ylpiperazin-1-yl)ethyl]quinolin-1(2H)-yl}acetamide

see trelanserin (INN)

2934 99 90

134379-77-4

4-amino-5-fluoro-1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]pyrimidin-2(1H)-one

see dexelvucitabine (INN)

2934 99 90

518048-05-0

potassium 4-[N-(2-fluorobenzyl)carbamoyl]-1-methyl-2-[1-methyl-1-(5-methyl-1,3,4-oxadiazole-2-carboxamido)ethyl]-6-oxo-1,6-dihydropyrimidine-5-olate

see raltegravir (INN)

2935 00 90

170569-88-7

4-[5-(4-fluorophenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzene-1-sulfonamide

see mavacoxib (INN)

2935 00 90

186497-07-4

N-(3-methoxy-5-methylpyrazin-2-yl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]pyridine-3-sulfonamide

see zibotentan (INN)